Future Oncology FEBRUARY 08, 2019

KEYNOTE-590: Phase III study of first-line chemotherapy with or without pembrolizumab for advanced esophageal cancer

Ken Kato, Manish A. Shah, Peter Enzinger, et al.

Bottom Line

The KEYNOTE-590 trial demonstrated that the addition of pembrolizumab to standard-of-care platinum-based chemotherapy significantly improves overall and progression-free survival in patients with previously untreated advanced or metastatic esophageal and esophagogastric junction (EGJ) cancers, regardless of histology or PD-L1 status.

Key Findings

1. In the overall intent-to-treat population, pembrolizumab plus chemotherapy significantly improved overall survival compared to placebo plus chemotherapy (median OS: 12.3 months vs. 9.8 months; hazard ratio [HR] 0.72; 95% CI, 0.62–0.84).
2. Long-term 5-year follow-up data indicated a persistent survival benefit, with an estimated 5-year survival rate of 10.6% in the pembrolizumab plus chemotherapy arm compared to 3.0% in the placebo plus chemotherapy arm.
3. Progression-free survival was significantly improved with the addition of pembrolizumab (median PFS: 6.3 months vs. 5.8 months; HR 0.65; 95% CI, 0.55–0.76).
4. Superiority was particularly pronounced in patients with esophageal squamous cell carcinoma and PD-L1 combined positive score (CPS) ≥10, where the median OS was 13.9 months with pembrolizumab plus chemotherapy compared to 8.8 months with placebo plus chemotherapy (HR 0.57; 95% CI, 0.43–0.75).
5. The addition of pembrolizumab was associated with a manageable safety profile, with no significant increase in treatment-related adverse events compared to chemotherapy alone.

Study Design

Design
RCT
Double-Blind
Sample
749
Patients
Duration
58.8 mo
Median
Setting
Multicenter, global
Population Patients with previously untreated, locally advanced, unresectable or metastatic adenocarcinoma or squamous cell carcinoma of the esophagus, or advanced/metastatic Siewert type 1 adenocarcinoma of the esophagogastric junction.
Intervention Pembrolizumab 200 mg every 3 weeks for up to 35 cycles, in combination with cisplatin (80 mg/m2 every 3 weeks) and 5-fluorouracil (800 mg/m2 per day on days 1–5 every 3 weeks).
Comparator Placebo plus cisplatin (80 mg/m2 every 3 weeks) and 5-fluorouracil (800 mg/m2 per day on days 1–5 every 3 weeks).
Outcome Overall survival and progression-free survival as assessed by investigator per RECIST v1.1.

Study Limitations

The study included a heterogeneous patient population (both adenocarcinoma and squamous cell carcinoma), which may complicate direct clinical application across distinct tumor histologies.
The absolute gain in median progression-free survival was relatively modest (0.5 months), despite achieving statistical significance.
Treatment-related toxicities, while manageable, increased with the addition of immunotherapy, necessitating close monitoring of immune-related adverse events.
The study excluded patients with performance status ≥2, limiting the generalizability of these findings to a broader, potentially more comorbid real-world population.

Clinical Significance

KEYNOTE-590 established the combination of pembrolizumab with platinum- and fluoropyrimidine-based chemotherapy as a new global standard of care for the first-line treatment of advanced or metastatic esophageal and Siewert type 1 EGJ carcinoma, demonstrating both a statistically significant and clinically meaningful improvement in long-term survival outcomes.

Historical Context

Prior to KEYNOTE-590, standard first-line therapy for advanced esophageal cancer was limited to platinum/fluoropyrimidine-based chemotherapy, which provided only modest survival benefits and carried a poor prognosis. The success of this trial represented a transformative shift in the treatment landscape by successfully integrating immune checkpoint inhibition into the frontline setting.

Guided Discussion

High-yield insights from every perspective

Med Student
Medical Student

What is the physiological mechanism by which pembrolizumab enhances the anti-tumor response in patients with advanced esophageal cancer, and why is this often combined with chemotherapy?

Key Response

Pembrolizumab is a monoclonal antibody that blocks the PD-1 receptor on T-cells, preventing it from binding to ligands PD-L1 and PD-L2 on tumor cells. This disruption prevents the 'off signal' that tumors use to evade the immune system. Chemotherapy is added because it can induce immunogenic cell death, releasing tumor antigens and potentially sensitizing the tumor microenvironment to immunotherapy, thereby creating a synergistic effect.

Resident
Resident

Based on the KEYNOTE-590 results, which specific patient subgroups demonstrated the most significant overall survival benefit, and how does this influence your initial workup for a newly diagnosed metastatic esophageal cancer patient?

Key Response

While KEYNOTE-590 showed benefit in the all-comer population, the most pronounced survival benefits were seen in patients with Esophageal Squamous Cell Carcinoma (ESCC) and those with a PD-L1 Combined Positive Score (CPS) ≥ 10. Consequently, the initial workup must include both histological confirmation and mandatory PD-L1 IHC testing to risk-stratify the patient and set expectations for the magnitude of treatment benefit.

Fellow
Fellow

Evaluate the clinical significance of the KEYNOTE-590 findings for patients with Esophageal Adenocarcinoma (EAC) versus Esophageal Squamous Cell Carcinoma (ESCC) in the context of competing data from trials like CheckMate 648.

Key Response

KEYNOTE-590 included both EAC and ESCC, demonstrating benefit across histologies, whereas CheckMate 648 focused strictly on ESCC. Fellows must recognize that while PD-1 inhibition is now a standard for both, the magnitude of benefit in EAC (often found at the EGJ) may be slightly less robust than in ESCC. In EAC, integration with HER2 status (per KEYNOTE-811) further complicates the first-line landscape, necessitating a nuanced approach to biomarker-driven therapy.

Attending
Attending

How does the transition to first-line chemo-immunotherapy for advanced esophageal cancer alter your management of treatment-related toxicities, specifically when differentiating between chemotherapy-induced mucositis and immune-related adverse events?

Key Response

The addition of pembrolizumab adds a layer of complexity to toxicity management. An Attending must lead the team in distinguishing between cisplatin-induced nephrotoxicity or 5-FU-induced diarrhea and immune-mediated colitis or nephritis. Prompt recognition of immune-related adverse events (irAEs) is vital, as they require steroids and potential cessation of the checkpoint inhibitor, rather than simple dose reductions or supportive care used for cytotoxic side effects.

Scholarly Review

Critical appraisal through the lens of expert reviewers and guideline development

PhD
PhD

Critique the hierarchical statistical testing strategy employed in KEYNOTE-590 and discuss how the multiplicity of primary endpoints (OS and PFS across various subgroups) affects the interpretation of the study's power and Type I error rate.

Key Response

KEYNOTE-590 used a complex gatekeeping procedure to control the family-wise error rate across multiple hypotheses (ESCC CPS ≥ 10, ESCC all, CPS ≥ 10 all, and all-randomized). This design is robust for regulatory approval but requires careful interpretation because the alpha is 'spent' across these groups. Researchers must consider whether the trial was truly powered for the smaller subsets or if the 'all-comer' benefit was driven primarily by the high-performing CPS ≥ 10 subgroup.

Journal Editor
Journal Editor

Assess the choice of 5-fluorouracil plus cisplatin as the control arm in KEYNOTE-590; does this choice limit the study's external validity in Western centers where FOLFOX is the preferred backbone?

Key Response

A critical reviewer would note that while 5-FU/Cisplatin was a global standard during trial design, many Western clinicians prefer FOLFOX due to its better tolerability profile (e.g., less emesis and nephrotoxicity). If the control arm is perceived as 'sub-optimal' or more toxic than current regional standards, it may slightly confound the perceived therapeutic index of the pembrolizumab-chemo combination, although subsequent data suggests the benefit of PD-1 inhibition is likely backbone-independent.

Guideline Committee
Guideline Committee

Considering the NCCN and ESMO guidelines, should pembrolizumab plus chemotherapy be recommended as a Category 1 preference for all patients with advanced esophageal cancer, or should it be restricted by CPS score?

Key Response

Current NCCN guidelines generally list pembrolizumab with chemotherapy as a Category 1 recommendation for first-line treatment. However, the strength of the recommendation is most robust for CPS ≥ 10. The committee must weigh the statistically significant OS benefit in the 'all-comer' group against the clinical meaningfulness of the benefit in the CPS < 1 population, where the hazard ratio often approaches 1.0, to decide if a 'preferred' status should be restricted to high-expressors.

Clinical Landscape

Noteworthy Related Trials

2019

ATTRACTION-3

n = 419 · Lancet Oncol

Tested

Nivolumab

Population

Patients with unresectable advanced or recurrent esophageal squamous-cell carcinoma refractory or intolerant to previous fluoropyrimidine and platinum-based chemotherapy

Comparator

Taxane chemotherapy (docetaxel or paclitaxel)

Endpoint

Overall survival

Key result: Nivolumab significantly improved overall survival compared with taxane chemotherapy in the second-line setting for advanced esophageal squamous-cell carcinoma.
2021

CheckMate 649

n = 1581 · Lancet

Tested

Nivolumab plus chemotherapy

Population

Patients with previously untreated advanced or metastatic gastric or gastro-oesophageal junction cancer

Comparator

Chemotherapy alone

Endpoint

Overall survival and progression-free survival

Key result: Nivolumab combined with chemotherapy resulted in significantly longer overall and progression-free survival compared with chemotherapy alone in patients with PD-L1 combined positive score of 5 or more.
2021

ESCORT-1st

n = 596 · JAMA

Tested

Camrelizumab plus chemotherapy

Population

Patients with untreated advanced esophageal squamous cell carcinoma

Comparator

Placebo plus chemotherapy

Endpoint

Overall survival and progression-free survival

Key result: Camrelizumab plus chemotherapy significantly improved overall survival and progression-free survival compared with placebo plus chemotherapy.

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